Regulator

Summary of regulator annotations and link-out to annotation databases

Basic gene annotations are collected from Uniprot and displayed with links to original sources. A quick link to explore the genomic context with Uniprot Browser is available.

ZNF282 - zinc finger protein 282

Function

Binds to the U5 repressive element (U5RE) of the human T cell leukemia virus type I long terminal repeat. It recognizes the 5'-TCCACCCC-3' sequence as a core motif and exerts a strong repressive effect on HTLV-I LTR-mediated expression.

Uniprot Browser
Entrez IDEnsEMBL IDPreferred NameUniprot ID
8427 ENSG00000170265 ZNF282 Q9UDV7

List of causal flows containing the regulator.

Causal Flows are statistically significant links between putative causal events (somatic mutations, copy number variations, chromosomal translocations, etc.) and the activity levels of regulators and regulons. In the causal flow, a mutation may causally activate or deactivate a downstream regulator which then might up- down-regulates a regulonthat contains genes with similar expression profiles and binding sites.

Causal Mechanistic Flows with ENSG00000170265 as Regulator

IDMutationRoleRegulatorRoleRegulon# downstream regulons# diffexp regulonsDrugs
CMF-07545ANO7down-regulatesZNF282activatesR-120541Drugs (112)

Regulator Drugs (0)

Regulon Drugs (112)

PROMETHAZINE HYDROCHLORIDE, TRIPROLIDINE, LEVOCETIRIZINE DIHYDROCHLORIDE, KETOTIFEN FUMARATE, PAZOPANIB, PYRILAMINE MALEATE, TRIPELENNAMINE, RUPATADINE, DOXYLAMINE SUCCINATE, PEMIGATINIB, BRIVANIB ALANINATE, MECLIZINE, ERDAFITINIB, BEPOTASTINE, BROMPHENIRAMINE, CLEMASTINE, OLOPATADINE HYDROCHLORIDE, CYPROHEPTADINE HYDROCHLORIDE, EPINASTINE HYDROCHLORIDE, TERFENADINE, CARBINOXAMINE MALEATE, DEXCHLORPHENIRAMINE, ORPHENADRINE HYDROCHLORIDE, HMPL-453, CHLORPHENIRAMINE MALEATE, DEXBROMPHENIRAMINE, OLOPATADINE, ASTEMIZOLE, CHLORPHENIRAMINE, HISTAMINE, PAZOPANIB HYDROCHLORIDE, LEVOCABASTINE, BRIVANIB, DEXBROMPHENIRAMINE MALEATE, EBASTINE, NINTEDANIB ESYLATE, CINNARIZINE, ABX-464, HYDROXYZINE, LORATADINE, LY2624803, PHENIRAMINE MALEATE, TRIPROLIDINE HYDROCHLORIDE, XL-999, DIPHENHYDRAMINE HYDROCHLORIDE, TRIMIPRAMINE, DOVITINIB, ROGARATINIB, BUCLIZINE, EPINASTINE, AZD-4547, ORPHENADRINE, ENMD-2076, KETOTIFEN, FEXOFENADINE, BILASTINE, INFIGRATINIB, FGFR INHIBITOR DEBIO 1347, CHLORPHENOXAMINE, LEVOCABASTINE HYDROCHLORIDE, DIBENZEPIN, PROMETHAZINE, INFIGRATINIB PHOSPHATE, AZELASTINE, DIPHENHYDRAMINE CITRATE, TOLAZOLINE, METHYLPROMAZINE, NINTEDANIB, AZELASTINE HYDROCHLORIDE, ANTAZOLINE, FUTIBATINIB, MASITINIB, CYCLIZINE, FEXOFENADINE HYDROCHLORIDE, DOXYLAMINE, CETIRIZINE HYDROCHLORIDE, DIPHENYLPYRALINE, ESMIRTAZAPINE MALEATE, ORANTINIB, LEVOCETIRIZINE, ACRIVASTINE, BEPOTASTINE BESYLATE, DIPHENHYDRAMINE, THENALIDINE, DIMENHYDRINATE, GSK-1004723, PYRILAMINE, ORPHENADRINE CITRATE, DEXCHLORPHENIRAMINE MALEATE, CYPROHEPTADINE, PHENIRAMINE, CLEMASTINE FUMARATE, OCRIPLASMIN, BROMODIPHENHYDRAMINE, DIMETHINDENE, AZATADINE, ESMIRTAZAPINE, BROMPHENIRAMINE MALEATE, MECLIZINE HYDROCHLORIDE, METHAPYRILENE, EMEDASTINE, MIZOLASTINE, DERAZANTINIB, E-7090, HYDROXYZINE PAMOATE, ALCAFTADINE, BETAHISTINE, CARBINOXAMINE, DESLORATADINE, CETIRIZINE, ENMD-981693, METHDILAZINE

CMF-09764MTF1up-regulatesZNF282activatesR-120542Drugs (112)

Regulator Drugs (0)

Regulon Drugs (112)

PROMETHAZINE HYDROCHLORIDE, TRIPROLIDINE, LEVOCETIRIZINE DIHYDROCHLORIDE, KETOTIFEN FUMARATE, PAZOPANIB, PYRILAMINE MALEATE, TRIPELENNAMINE, RUPATADINE, DOXYLAMINE SUCCINATE, PEMIGATINIB, BRIVANIB ALANINATE, MECLIZINE, ERDAFITINIB, BEPOTASTINE, BROMPHENIRAMINE, CLEMASTINE, OLOPATADINE HYDROCHLORIDE, CYPROHEPTADINE HYDROCHLORIDE, EPINASTINE HYDROCHLORIDE, TERFENADINE, CARBINOXAMINE MALEATE, DEXCHLORPHENIRAMINE, ORPHENADRINE HYDROCHLORIDE, HMPL-453, CHLORPHENIRAMINE MALEATE, DEXBROMPHENIRAMINE, OLOPATADINE, ASTEMIZOLE, CHLORPHENIRAMINE, HISTAMINE, PAZOPANIB HYDROCHLORIDE, LEVOCABASTINE, BRIVANIB, DEXBROMPHENIRAMINE MALEATE, EBASTINE, NINTEDANIB ESYLATE, CINNARIZINE, ABX-464, HYDROXYZINE, LORATADINE, LY2624803, PHENIRAMINE MALEATE, TRIPROLIDINE HYDROCHLORIDE, XL-999, DIPHENHYDRAMINE HYDROCHLORIDE, TRIMIPRAMINE, DOVITINIB, ROGARATINIB, BUCLIZINE, EPINASTINE, AZD-4547, ORPHENADRINE, ENMD-2076, KETOTIFEN, FEXOFENADINE, BILASTINE, INFIGRATINIB, FGFR INHIBITOR DEBIO 1347, CHLORPHENOXAMINE, LEVOCABASTINE HYDROCHLORIDE, DIBENZEPIN, PROMETHAZINE, INFIGRATINIB PHOSPHATE, AZELASTINE, DIPHENHYDRAMINE CITRATE, TOLAZOLINE, METHYLPROMAZINE, NINTEDANIB, AZELASTINE HYDROCHLORIDE, ANTAZOLINE, FUTIBATINIB, MASITINIB, CYCLIZINE, FEXOFENADINE HYDROCHLORIDE, DOXYLAMINE, CETIRIZINE HYDROCHLORIDE, DIPHENYLPYRALINE, ESMIRTAZAPINE MALEATE, ORANTINIB, LEVOCETIRIZINE, ACRIVASTINE, BEPOTASTINE BESYLATE, DIPHENHYDRAMINE, THENALIDINE, DIMENHYDRINATE, GSK-1004723, PYRILAMINE, ORPHENADRINE CITRATE, DEXCHLORPHENIRAMINE MALEATE, CYPROHEPTADINE, PHENIRAMINE, CLEMASTINE FUMARATE, OCRIPLASMIN, BROMODIPHENHYDRAMINE, DIMETHINDENE, AZATADINE, ESMIRTAZAPINE, BROMPHENIRAMINE MALEATE, MECLIZINE HYDROCHLORIDE, METHAPYRILENE, EMEDASTINE, MIZOLASTINE, DERAZANTINIB, E-7090, HYDROXYZINE PAMOATE, ALCAFTADINE, BETAHISTINE, CARBINOXAMINE, DESLORATADINE, CETIRIZINE, ENMD-981693, METHDILAZINE

CMF-12092NOX3up-regulatesZNF282activatesR-120541Drugs (112)

Regulator Drugs (0)

Regulon Drugs (112)

PROMETHAZINE HYDROCHLORIDE, TRIPROLIDINE, LEVOCETIRIZINE DIHYDROCHLORIDE, KETOTIFEN FUMARATE, PAZOPANIB, PYRILAMINE MALEATE, TRIPELENNAMINE, RUPATADINE, DOXYLAMINE SUCCINATE, PEMIGATINIB, BRIVANIB ALANINATE, MECLIZINE, ERDAFITINIB, BEPOTASTINE, BROMPHENIRAMINE, CLEMASTINE, OLOPATADINE HYDROCHLORIDE, CYPROHEPTADINE HYDROCHLORIDE, EPINASTINE HYDROCHLORIDE, TERFENADINE, CARBINOXAMINE MALEATE, DEXCHLORPHENIRAMINE, ORPHENADRINE HYDROCHLORIDE, HMPL-453, CHLORPHENIRAMINE MALEATE, DEXBROMPHENIRAMINE, OLOPATADINE, ASTEMIZOLE, CHLORPHENIRAMINE, HISTAMINE, PAZOPANIB HYDROCHLORIDE, LEVOCABASTINE, BRIVANIB, DEXBROMPHENIRAMINE MALEATE, EBASTINE, NINTEDANIB ESYLATE, CINNARIZINE, ABX-464, HYDROXYZINE, LORATADINE, LY2624803, PHENIRAMINE MALEATE, TRIPROLIDINE HYDROCHLORIDE, XL-999, DIPHENHYDRAMINE HYDROCHLORIDE, TRIMIPRAMINE, DOVITINIB, ROGARATINIB, BUCLIZINE, EPINASTINE, AZD-4547, ORPHENADRINE, ENMD-2076, KETOTIFEN, FEXOFENADINE, BILASTINE, INFIGRATINIB, FGFR INHIBITOR DEBIO 1347, CHLORPHENOXAMINE, LEVOCABASTINE HYDROCHLORIDE, DIBENZEPIN, PROMETHAZINE, INFIGRATINIB PHOSPHATE, AZELASTINE, DIPHENHYDRAMINE CITRATE, TOLAZOLINE, METHYLPROMAZINE, NINTEDANIB, AZELASTINE HYDROCHLORIDE, ANTAZOLINE, FUTIBATINIB, MASITINIB, CYCLIZINE, FEXOFENADINE HYDROCHLORIDE, DOXYLAMINE, CETIRIZINE HYDROCHLORIDE, DIPHENYLPYRALINE, ESMIRTAZAPINE MALEATE, ORANTINIB, LEVOCETIRIZINE, ACRIVASTINE, BEPOTASTINE BESYLATE, DIPHENHYDRAMINE, THENALIDINE, DIMENHYDRINATE, GSK-1004723, PYRILAMINE, ORPHENADRINE CITRATE, DEXCHLORPHENIRAMINE MALEATE, CYPROHEPTADINE, PHENIRAMINE, CLEMASTINE FUMARATE, OCRIPLASMIN, BROMODIPHENHYDRAMINE, DIMETHINDENE, AZATADINE, ESMIRTAZAPINE, BROMPHENIRAMINE MALEATE, MECLIZINE HYDROCHLORIDE, METHAPYRILENE, EMEDASTINE, MIZOLASTINE, DERAZANTINIB, E-7090, HYDROXYZINE PAMOATE, ALCAFTADINE, BETAHISTINE, CARBINOXAMINE, DESLORATADINE, CETIRIZINE, ENMD-981693, METHDILAZINE

CMF-14949SDHAP3up-regulatesZNF282activatesR-120541Drugs (112)

Regulator Drugs (0)

Regulon Drugs (112)

PROMETHAZINE HYDROCHLORIDE, TRIPROLIDINE, LEVOCETIRIZINE DIHYDROCHLORIDE, KETOTIFEN FUMARATE, PAZOPANIB, PYRILAMINE MALEATE, TRIPELENNAMINE, RUPATADINE, DOXYLAMINE SUCCINATE, PEMIGATINIB, BRIVANIB ALANINATE, MECLIZINE, ERDAFITINIB, BEPOTASTINE, BROMPHENIRAMINE, CLEMASTINE, OLOPATADINE HYDROCHLORIDE, CYPROHEPTADINE HYDROCHLORIDE, EPINASTINE HYDROCHLORIDE, TERFENADINE, CARBINOXAMINE MALEATE, DEXCHLORPHENIRAMINE, ORPHENADRINE HYDROCHLORIDE, HMPL-453, CHLORPHENIRAMINE MALEATE, DEXBROMPHENIRAMINE, OLOPATADINE, ASTEMIZOLE, CHLORPHENIRAMINE, HISTAMINE, PAZOPANIB HYDROCHLORIDE, LEVOCABASTINE, BRIVANIB, DEXBROMPHENIRAMINE MALEATE, EBASTINE, NINTEDANIB ESYLATE, CINNARIZINE, ABX-464, HYDROXYZINE, LORATADINE, LY2624803, PHENIRAMINE MALEATE, TRIPROLIDINE HYDROCHLORIDE, XL-999, DIPHENHYDRAMINE HYDROCHLORIDE, TRIMIPRAMINE, DOVITINIB, ROGARATINIB, BUCLIZINE, EPINASTINE, AZD-4547, ORPHENADRINE, ENMD-2076, KETOTIFEN, FEXOFENADINE, BILASTINE, INFIGRATINIB, FGFR INHIBITOR DEBIO 1347, CHLORPHENOXAMINE, LEVOCABASTINE HYDROCHLORIDE, DIBENZEPIN, PROMETHAZINE, INFIGRATINIB PHOSPHATE, AZELASTINE, DIPHENHYDRAMINE CITRATE, TOLAZOLINE, METHYLPROMAZINE, NINTEDANIB, AZELASTINE HYDROCHLORIDE, ANTAZOLINE, FUTIBATINIB, MASITINIB, CYCLIZINE, FEXOFENADINE HYDROCHLORIDE, DOXYLAMINE, CETIRIZINE HYDROCHLORIDE, DIPHENYLPYRALINE, ESMIRTAZAPINE MALEATE, ORANTINIB, LEVOCETIRIZINE, ACRIVASTINE, BEPOTASTINE BESYLATE, DIPHENHYDRAMINE, THENALIDINE, DIMENHYDRINATE, GSK-1004723, PYRILAMINE, ORPHENADRINE CITRATE, DEXCHLORPHENIRAMINE MALEATE, CYPROHEPTADINE, PHENIRAMINE, CLEMASTINE FUMARATE, OCRIPLASMIN, BROMODIPHENHYDRAMINE, DIMETHINDENE, AZATADINE, ESMIRTAZAPINE, BROMPHENIRAMINE MALEATE, MECLIZINE HYDROCHLORIDE, METHAPYRILENE, EMEDASTINE, MIZOLASTINE, DERAZANTINIB, E-7090, HYDROXYZINE PAMOATE, ALCAFTADINE, BETAHISTINE, CARBINOXAMINE, DESLORATADINE, CETIRIZINE, ENMD-981693, METHDILAZINE

CMF-15193ERCC6down-regulatesZNF282activatesR-120541Drugs (112)

Regulator Drugs (0)

Regulon Drugs (112)

PROMETHAZINE HYDROCHLORIDE, TRIPROLIDINE, LEVOCETIRIZINE DIHYDROCHLORIDE, KETOTIFEN FUMARATE, PAZOPANIB, PYRILAMINE MALEATE, TRIPELENNAMINE, RUPATADINE, DOXYLAMINE SUCCINATE, PEMIGATINIB, BRIVANIB ALANINATE, MECLIZINE, ERDAFITINIB, BEPOTASTINE, BROMPHENIRAMINE, CLEMASTINE, OLOPATADINE HYDROCHLORIDE, CYPROHEPTADINE HYDROCHLORIDE, EPINASTINE HYDROCHLORIDE, TERFENADINE, CARBINOXAMINE MALEATE, DEXCHLORPHENIRAMINE, ORPHENADRINE HYDROCHLORIDE, HMPL-453, CHLORPHENIRAMINE MALEATE, DEXBROMPHENIRAMINE, OLOPATADINE, ASTEMIZOLE, CHLORPHENIRAMINE, HISTAMINE, PAZOPANIB HYDROCHLORIDE, LEVOCABASTINE, BRIVANIB, DEXBROMPHENIRAMINE MALEATE, EBASTINE, NINTEDANIB ESYLATE, CINNARIZINE, ABX-464, HYDROXYZINE, LORATADINE, LY2624803, PHENIRAMINE MALEATE, TRIPROLIDINE HYDROCHLORIDE, XL-999, DIPHENHYDRAMINE HYDROCHLORIDE, TRIMIPRAMINE, DOVITINIB, ROGARATINIB, BUCLIZINE, EPINASTINE, AZD-4547, ORPHENADRINE, ENMD-2076, KETOTIFEN, FEXOFENADINE, BILASTINE, INFIGRATINIB, FGFR INHIBITOR DEBIO 1347, CHLORPHENOXAMINE, LEVOCABASTINE HYDROCHLORIDE, DIBENZEPIN, PROMETHAZINE, INFIGRATINIB PHOSPHATE, AZELASTINE, DIPHENHYDRAMINE CITRATE, TOLAZOLINE, METHYLPROMAZINE, NINTEDANIB, AZELASTINE HYDROCHLORIDE, ANTAZOLINE, FUTIBATINIB, MASITINIB, CYCLIZINE, FEXOFENADINE HYDROCHLORIDE, DOXYLAMINE, CETIRIZINE HYDROCHLORIDE, DIPHENYLPYRALINE, ESMIRTAZAPINE MALEATE, ORANTINIB, LEVOCETIRIZINE, ACRIVASTINE, BEPOTASTINE BESYLATE, DIPHENHYDRAMINE, THENALIDINE, DIMENHYDRINATE, GSK-1004723, PYRILAMINE, ORPHENADRINE CITRATE, DEXCHLORPHENIRAMINE MALEATE, CYPROHEPTADINE, PHENIRAMINE, CLEMASTINE FUMARATE, OCRIPLASMIN, BROMODIPHENHYDRAMINE, DIMETHINDENE, AZATADINE, ESMIRTAZAPINE, BROMPHENIRAMINE MALEATE, MECLIZINE HYDROCHLORIDE, METHAPYRILENE, EMEDASTINE, MIZOLASTINE, DERAZANTINIB, E-7090, HYDROXYZINE PAMOATE, ALCAFTADINE, BETAHISTINE, CARBINOXAMINE, DESLORATADINE, CETIRIZINE, ENMD-981693, METHDILAZINE

CMF-21413GRIK3up-regulatesZNF282activatesR-120541Drugs (112)

Regulator Drugs (0)

Regulon Drugs (112)

PROMETHAZINE HYDROCHLORIDE, TRIPROLIDINE, LEVOCETIRIZINE DIHYDROCHLORIDE, KETOTIFEN FUMARATE, PAZOPANIB, PYRILAMINE MALEATE, TRIPELENNAMINE, RUPATADINE, DOXYLAMINE SUCCINATE, PEMIGATINIB, BRIVANIB ALANINATE, MECLIZINE, ERDAFITINIB, BEPOTASTINE, BROMPHENIRAMINE, CLEMASTINE, OLOPATADINE HYDROCHLORIDE, CYPROHEPTADINE HYDROCHLORIDE, EPINASTINE HYDROCHLORIDE, TERFENADINE, CARBINOXAMINE MALEATE, DEXCHLORPHENIRAMINE, ORPHENADRINE HYDROCHLORIDE, HMPL-453, CHLORPHENIRAMINE MALEATE, DEXBROMPHENIRAMINE, OLOPATADINE, ASTEMIZOLE, CHLORPHENIRAMINE, HISTAMINE, PAZOPANIB HYDROCHLORIDE, LEVOCABASTINE, BRIVANIB, DEXBROMPHENIRAMINE MALEATE, EBASTINE, NINTEDANIB ESYLATE, CINNARIZINE, ABX-464, HYDROXYZINE, LORATADINE, LY2624803, PHENIRAMINE MALEATE, TRIPROLIDINE HYDROCHLORIDE, XL-999, DIPHENHYDRAMINE HYDROCHLORIDE, TRIMIPRAMINE, DOVITINIB, ROGARATINIB, BUCLIZINE, EPINASTINE, AZD-4547, ORPHENADRINE, ENMD-2076, KETOTIFEN, FEXOFENADINE, BILASTINE, INFIGRATINIB, FGFR INHIBITOR DEBIO 1347, CHLORPHENOXAMINE, LEVOCABASTINE HYDROCHLORIDE, DIBENZEPIN, PROMETHAZINE, INFIGRATINIB PHOSPHATE, AZELASTINE, DIPHENHYDRAMINE CITRATE, TOLAZOLINE, METHYLPROMAZINE, NINTEDANIB, AZELASTINE HYDROCHLORIDE, ANTAZOLINE, FUTIBATINIB, MASITINIB, CYCLIZINE, FEXOFENADINE HYDROCHLORIDE, DOXYLAMINE, CETIRIZINE HYDROCHLORIDE, DIPHENYLPYRALINE, ESMIRTAZAPINE MALEATE, ORANTINIB, LEVOCETIRIZINE, ACRIVASTINE, BEPOTASTINE BESYLATE, DIPHENHYDRAMINE, THENALIDINE, DIMENHYDRINATE, GSK-1004723, PYRILAMINE, ORPHENADRINE CITRATE, DEXCHLORPHENIRAMINE MALEATE, CYPROHEPTADINE, PHENIRAMINE, CLEMASTINE FUMARATE, OCRIPLASMIN, BROMODIPHENHYDRAMINE, DIMETHINDENE, AZATADINE, ESMIRTAZAPINE, BROMPHENIRAMINE MALEATE, MECLIZINE HYDROCHLORIDE, METHAPYRILENE, EMEDASTINE, MIZOLASTINE, DERAZANTINIB, E-7090, HYDROXYZINE PAMOATE, ALCAFTADINE, BETAHISTINE, CARBINOXAMINE, DESLORATADINE, CETIRIZINE, ENMD-981693, METHDILAZINE

CMF-25079IQSEC3up-regulatesZNF282activatesR-120543Drugs (112)

Regulator Drugs (0)

Regulon Drugs (112)

PROMETHAZINE HYDROCHLORIDE, TRIPROLIDINE, LEVOCETIRIZINE DIHYDROCHLORIDE, KETOTIFEN FUMARATE, PAZOPANIB, PYRILAMINE MALEATE, TRIPELENNAMINE, RUPATADINE, DOXYLAMINE SUCCINATE, PEMIGATINIB, BRIVANIB ALANINATE, MECLIZINE, ERDAFITINIB, BEPOTASTINE, BROMPHENIRAMINE, CLEMASTINE, OLOPATADINE HYDROCHLORIDE, CYPROHEPTADINE HYDROCHLORIDE, EPINASTINE HYDROCHLORIDE, TERFENADINE, CARBINOXAMINE MALEATE, DEXCHLORPHENIRAMINE, ORPHENADRINE HYDROCHLORIDE, HMPL-453, CHLORPHENIRAMINE MALEATE, DEXBROMPHENIRAMINE, OLOPATADINE, ASTEMIZOLE, CHLORPHENIRAMINE, HISTAMINE, PAZOPANIB HYDROCHLORIDE, LEVOCABASTINE, BRIVANIB, DEXBROMPHENIRAMINE MALEATE, EBASTINE, NINTEDANIB ESYLATE, CINNARIZINE, ABX-464, HYDROXYZINE, LORATADINE, LY2624803, PHENIRAMINE MALEATE, TRIPROLIDINE HYDROCHLORIDE, XL-999, DIPHENHYDRAMINE HYDROCHLORIDE, TRIMIPRAMINE, DOVITINIB, ROGARATINIB, BUCLIZINE, EPINASTINE, AZD-4547, ORPHENADRINE, ENMD-2076, KETOTIFEN, FEXOFENADINE, BILASTINE, INFIGRATINIB, FGFR INHIBITOR DEBIO 1347, CHLORPHENOXAMINE, LEVOCABASTINE HYDROCHLORIDE, DIBENZEPIN, PROMETHAZINE, INFIGRATINIB PHOSPHATE, AZELASTINE, DIPHENHYDRAMINE CITRATE, TOLAZOLINE, METHYLPROMAZINE, NINTEDANIB, AZELASTINE HYDROCHLORIDE, ANTAZOLINE, FUTIBATINIB, MASITINIB, CYCLIZINE, FEXOFENADINE HYDROCHLORIDE, DOXYLAMINE, CETIRIZINE HYDROCHLORIDE, DIPHENYLPYRALINE, ESMIRTAZAPINE MALEATE, ORANTINIB, LEVOCETIRIZINE, ACRIVASTINE, BEPOTASTINE BESYLATE, DIPHENHYDRAMINE, THENALIDINE, DIMENHYDRINATE, GSK-1004723, PYRILAMINE, ORPHENADRINE CITRATE, DEXCHLORPHENIRAMINE MALEATE, CYPROHEPTADINE, PHENIRAMINE, CLEMASTINE FUMARATE, OCRIPLASMIN, BROMODIPHENHYDRAMINE, DIMETHINDENE, AZATADINE, ESMIRTAZAPINE, BROMPHENIRAMINE MALEATE, MECLIZINE HYDROCHLORIDE, METHAPYRILENE, EMEDASTINE, MIZOLASTINE, DERAZANTINIB, E-7090, HYDROXYZINE PAMOATE, ALCAFTADINE, BETAHISTINE, CARBINOXAMINE, DESLORATADINE, CETIRIZINE, ENMD-981693, METHDILAZINE